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Accelerated structure-based design of chemically diverse allosteric modulators of a muscarinic G protein-coupled receptor
Yinglong Miao, Dahlia Anne Goldfeld, Ee Von Moo, Patrick M. Sexton, Arthur Christopoulos, J. Andrew McCammon, and Celine Valant
Yinglong Miao
aHoward Hughes Medical Institute, University of California at San Diego, La Jolla, CA 92093;bDepartment of Pharmacology, University of California at San Diego, La Jolla, CA 92093;
Dahlia Anne Goldfeld
bDepartment of Pharmacology, University of California at San Diego, La Jolla, CA 92093;
Ee Von Moo
cDrug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville VIC 3052, Australia;
Patrick M. Sexton
cDrug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville VIC 3052, Australia;
Arthur Christopoulos
cDrug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville VIC 3052, Australia;
J. Andrew McCammon
aHoward Hughes Medical Institute, University of California at San Diego, La Jolla, CA 92093;bDepartment of Pharmacology, University of California at San Diego, La Jolla, CA 92093;dDepartment of Chemistry and Biochemistry, University of California at San Diego, La Jolla, CA 92093
Celine Valant
cDrug Discovery Biology, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville VIC 3052, Australia;